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More on Pharmaceuticals and Intermediates

 

Pharmaceuticals and Intermediates - Products

 

Intermediates: Phosgene Derivatives
Product CAS No. Application
Chloroformates
1-Chloroethyl Chloroformate 50893-53-3 Ampiroxicam, Candesartan
2,2,2-Trichloroethyl Chloroformate 17341-93-4 Cabergoline, Naltrexone, Nalbuphine
Isobutyl Chloroformate 543-27-1 Mosapride, Nelfinavir, Phenethicillin
4-Nitro Benzyl Chloroformate 4457-32-3 Meropenem, Panipenem, Biapenem
4-Nitro Phenyl Chloroformate 7693-46-1 Ritonavir, Efavirenz, Pibrozelesin
Phenyl Chloroformate 1885-14-9 Camazepam, Itraconazole, Paroxetin
n-Pentyl Chlorformate 638-41-5 Capacitabine
Isocyanates
Cyclohexyl Isocyanate * 3173-53-3 Glibenclamide, Glipizide, Glycyclamide
2-Phenyl Ethyl Isocyanate 1943-82-4 Glimepiride
Para Toluene Sulfonyl Isocyanate 4083-64-1 Coating Application
Phenyl Isocyanate 103-71-9 Devazepid
NCA
Z-L-Valine NCA 158257-41-1 Valganciclovir
N6-(trifluroacetyl)_N2-Carboxy-L-Lysine anhydride *   Lisinopril
Carbonate & Dicarbonate
1-Chloro Ethyl Isopropyl Carbonate 98298-66-9 Cefpodoxime proxetil, Bacampicillin
1-Chloro Ethyl Cyclohexyl Carbonate 99464-83-2 Cefotiam Hexetil (SCE-2174),TCV-116
Di-tert-butyl Dicarbonate (Di-BOC)* 24424-99-5 Fosinopril, Nevirapine
Chloride
N'-Methyl piperazine carbamoyl chloride.HCl 55112-42-0 Zopiclone
Vilsmeier reagent 3724-43-4 Formylation, Dehydration & Chlorination
Ureas
N,N'-Carbonyl diimidazole (CDI) 530-62-1 Meropenem, Nebivolol, Sildenafil
Tetra Butyl Ureas ( TBU ) 4559-86-8 Catalyst
Others
(R) - (+)-a, a – Diphenyl Prolinol 22348-32-9 Treprostinil, Ezetimibe
(S)- (-) - a, a – Diphenyl Prolinol 112068-01-6 (S)-Salmeterol
L-Prolinamide 7531-52-4 Montirelin, Posatirelin, Protirelin



Bulk Actives
Product CAS No. Application
Acyclovir USP 59277-89-3 Anti-Viral
Dapsone 80-08-0 Anti-Bacterial
Roxithromycin EP 80214-83-1 Anti-Bacterial
Bethanechol chloride USP * 590-63-6 Cholinergic



Bulk Chemicals
Product CAS No. Application
4,4'-Diamino Diphenyl Sulphone 80-08-0 Epoxy Hardner,Aerospace Industry, Laminates Industry
3,3'-Diamino Diphenyl Sulphone 599-61-1 Epoxy Hardner,Aerospace Industry, Laminates Industry
Ethyl-(4-toluene sulfonyl)-carbamate 5577-13-9 Veterinary Application
N,N'-Dibenzyl Ethylene Diamine Diacetate 122-75-8 Benzathine Penicilline



On Campaign Basis
Product CAS No. Application
Allyl Chloroformate 2937-50-0 Alloxycarbonyl Protection of Amines
N-BenzylOxy Carbonyl -L- Valine* 1149-26-4 Valaciclovir
Di - Isopropyl Hydrazo di Carboxylate 19740-72-8 Catalyst for Oxidation of alcohol
4-Fluoro Phenyl isocyanate 1195-45-5 Photographic chemical
Isopropyl Chloroformate 108-23-6 Altropane(1231), Doripenem, Opaviraline
1-Pyrrolidine Carbonyl Chloride 1192-63-8 New Drug Development
4-Methoxy Phenyl Chloroformate 7693-41-6 New Drug Development
Bis ( 4-Nitrophenyl ) Carbonate 5070-13-3 CI-1021, Ritonavir
2-Methoxyethyl chloroformate 628-12-6 New Drug Developments



Under Development
Product CAS No. Application
Oxalyl Chloride 79-37-8 Ezetimibe, Epresteride,Mecillinam
Bis(4-Methylbenzyl) peroxydicarbonate 53728-93-1 Flomoxef
Para Phenylene Diisocyanate 104-49-4 Polyurethane Application
t-4 Me Cyclohexyl Isocyanate 32175-00-1 Glimepiride
( R )-2-Methyl-CBS-Oxazaborolidine.H20 112022-83-0 Treprostinil, Ezetimibe

 

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